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Compound
PGDB_C027542
4 activity records2 related patents
2D structure
COc1ccc(-c2nnc(NC3CN(c4cc(F)c(C5CCC(=O)NC5=O)c(F)c4)C3)o2)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | > | 80 | % | 30 uM | 24 h | CDK2 | - | HEK293 | WO2025224262A1 | PGDB_A012797 | PGDB_C027542 | PGDB_AS001415 | View |
| Ki | - | <= | 0.1 | uM | - | — | - | - | - | WO2024092039 | PGDB_A028568 | PGDB_C027542 | PGDB_AS001899 | View |
| Dmax | - | > | 80 | % | 30 uM | 24 h | - | - | HEK293 | WO2024092039 | PGDB_A049677 | PGDB_C027542 | PGDB_AS002575 | View |
| Ki | - | <= | 0.1 | uM | - | — | CRBN | CRBN | - | WO2025224262A1 | PGDB_A074362 | PGDB_C027542 | PGDB_AS001844 | View |