Assay context summary

Assay context

52 activity records
Activity compounds and values

Activity records

52 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031991
IC50-=86nM--CRBNLS513WO2026114958A1PGDB_A000184PGDB_C031991PGDB_AS001452View
2D structure for PGDB_C031992
IC50-=11.3nM--CRBNLS513WO2026114958A1PGDB_A000288PGDB_C031992PGDB_AS001452View
2D structure for PGDB_C031950
IC50-=437.1nM--CRBNLS513WO2026114958A1PGDB_A000529PGDB_C031950PGDB_AS001452View
2D structure for PGDB_C031951
IC50-=25.8nM--CRBNLS513WO2026114958A1PGDB_A000564PGDB_C031951PGDB_AS001452View
2D structure for PGDB_C031993
IC50-=29.2nM--CRBNLS513WO2026114958A1PGDB_A000587PGDB_C031993PGDB_AS001452View
2D structure for PGDB_C031983
IC50-=394.8nM--CRBNLS513WO2026114958A1PGDB_A001328PGDB_C031983PGDB_AS001452View
2D structure for PGDB_C031969
IC50-=17.6nM--CRBNLS513WO2026114958A1PGDB_A001520PGDB_C031969PGDB_AS001452View
2D structure for PGDB_C031996
IC50-=6nM--CRBNLS513WO2026114958A1PGDB_A001545PGDB_C031996PGDB_AS001452View
2D structure for PGDB_C031949
IC50-=7.2nM--CRBNLS513WO2026114958A1PGDB_A001644PGDB_C031949PGDB_AS001452View
2D structure for PGDB_C031941
IC50-=8.3nM--CRBNLS513WO2026114958A1PGDB_A002602PGDB_C031941PGDB_AS001452View
2D structure for PGDB_C031980
IC50-=124.2nM--CRBNLS513WO2026114958A1PGDB_A003008PGDB_C031980PGDB_AS001452View
2D structure for PGDB_C031961
IC50-=134.1nM--CRBNLS513WO2026114958A1PGDB_A003040PGDB_C031961PGDB_AS001452View
2D structure for PGDB_C031959
IC50-=106.1nM--CRBNLS513WO2026114958A1PGDB_A003272PGDB_C031959PGDB_AS001452View
2D structure for PGDB_C031964
IC50-=44.6nM--CRBNLS513WO2026114958A1PGDB_A003284PGDB_C031964PGDB_AS001452View
2D structure for PGDB_C031947
IC50-=429.1nM--CRBNLS513WO2026114958A1PGDB_A003615PGDB_C031947PGDB_AS001452View
2D structure for PGDB_C031984
IC50-=34.2nM--CRBNLS513WO2026114958A1PGDB_A003713PGDB_C031984PGDB_AS001452View
2D structure for PGDB_C031957
IC50-=104.3nM--CRBNLS513WO2026114958A1PGDB_A003738PGDB_C031957PGDB_AS001452View
2D structure for PGDB_C031962
IC50-=252.1nM--CRBNLS513WO2026114958A1PGDB_A003854PGDB_C031962PGDB_AS001452View
2D structure for PGDB_C031956
IC50-=55.3nM--CRBNLS513WO2026114958A1PGDB_A003857PGDB_C031956PGDB_AS001452View
2D structure for PGDB_C031955
IC50-=64.3nM--CRBNLS513WO2026114958A1PGDB_A004388PGDB_C031955PGDB_AS001452View