Assay

PGDB_AS001495

System: cell_basedTarget: CRBN
Assay context summary

Assay context

9 activity records
Assay familybiochemical
Systemcell_based
ReadoutKd
TargetCRBN
E3CRBN
OrganismHomo sapiens
TechnologyHTRF
Activity compounds and values

Activity records

9 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C014203
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A012777PGDB_C014203PGDB_AS001495View
2D structure for PGDB_C014202
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A015441PGDB_C014202PGDB_AS001495View
2D structure for PGDB_C014200
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A015746PGDB_C014200PGDB_AS001495View
2D structure for PGDB_C023634
% Inhibition-=30-40%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A016867PGDB_C023634PGDB_AS001495View
2D structure for PGDB_C023631
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A022287PGDB_C023631PGDB_AS001495View
2D structure for PGDB_C023635
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A042654PGDB_C023635PGDB_AS001495View
2D structure for PGDB_C014201
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A057234PGDB_C014201PGDB_AS001495View
2D structure for PGDB_C023633
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A062302PGDB_C023633PGDB_AS001495View
2D structure for PGDB_C023632
% Inhibition-=20-30%0.5 uM3 hCRBNCRBN-WO2024245444A1PGDB_A070854PGDB_C023632PGDB_AS001495View
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