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CC(F)(F)c1ncc(NC(=O)NC2CN(c3cc(F)c(C4CCC(=O)NC4=O)c(F)c3)C2)cc1C#CC1CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 170.8 | nM | - | — | GSPT1 | - | ABC-1 | CN119264113A | PGDB_A042982 | PGDB_C000671 | PGDB_AS001474 | View | |
| IC50 | - | = | 68.9 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A061884 | PGDB_C000671 | PGDB_AS001498 | View | |
| DC50 | - | = | 219.2 | nM | - | — | GSPT1 | - | CAL-51 | CN119264113A | PGDB_A064642 | PGDB_C000671 | PGDB_AS001139 | View | |
| IC50 | - | = | 10 | nM | - | — | GSPT1 | - | ABC-1 | CN119264113A | PGDB_A076149 | PGDB_C000671 | PGDB_AS002488 | View |