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SIMM · NJU
Assay
PGDB_AS001553
System: cell_based
Target: NEK7
Assay context summary
Assay context
19 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
NEK7
E3
CRBN
Activity compounds and values
Activity records
19 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
26
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A008067
PGDB_C020455
PGDB_AS001553
View
Dmax
-
=
7
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A011286
PGDB_C020436
PGDB_AS001553
View
Dmax
-
=
33
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A013712
PGDB_C020449
PGDB_AS001553
View
Dmax
-
=
136
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A019958
PGDB_C020446
PGDB_AS001553
View
Dmax
-
=
672
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A026126
PGDB_C020452
PGDB_AS001553
View
Dmax
-
=
143
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A027078
PGDB_C020453
PGDB_AS001553
View
Dmax
-
=
12
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A027305
PGDB_C020435
PGDB_AS001553
View
Dmax
-
=
3
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A030117
PGDB_C020440
PGDB_AS001553
View
Dmax
-
=
15
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A037980
PGDB_C020439
PGDB_AS001553
View
Dmax
-
=
1000
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A038192
PGDB_C020447
PGDB_AS001553
View
Dmax
-
=
213
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A039361
PGDB_C020444
PGDB_AS001553
View
Dmax
-
=
11
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A039880
PGDB_C020438
PGDB_AS001553
View
Dmax
-
=
76
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A050007
PGDB_C020451
PGDB_AS001553
View
Dmax
-
=
155
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A050209
PGDB_C020450
PGDB_AS001553
View
Dmax
-
=
179
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A050728
PGDB_C020454
PGDB_AS001553
View
Dmax
-
=
1
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A051405
PGDB_C020442
PGDB_AS001553
View
Dmax
-
=
100
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057655
PGDB_C020437
PGDB_AS001553
View
Dmax
-
=
190
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057784
PGDB_C020448
PGDB_AS001553
View
Dmax
-
=
312
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A064330
PGDB_C020445
PGDB_AS001553
View