Assay

PGDB_AS001560

System: biochemicalTarget: CRBN
Assay context summary

Assay context

60 activity records
Assay familybinding
Systembiochemical
ReadoutIC50
TargetCRBN
E3CRBN
OrganismHomo sapiens
Activity compounds and values

Activity records

60 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C009809
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A008926PGDB_C009809PGDB_AS001560View
2D structure for PGDB_C009805
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A009117PGDB_C009805PGDB_AS001560View
2D structure for PGDB_C009825
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A009699PGDB_C009825PGDB_AS001560View
2D structure for PGDB_C009820
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A010916PGDB_C009820PGDB_AS001560View
2D structure for PGDB_C009821
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A011670PGDB_C009821PGDB_AS001560View
2D structure for PGDB_C009819
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A013774PGDB_C009819PGDB_AS001560View
2D structure for PGDB_C009804
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A014280PGDB_C009804PGDB_AS001560View
2D structure for PGDB_C009849
IC50-=0.5-1uM-—CRBNCRBN-WO2022187423A1PGDB_A014642PGDB_C009849PGDB_AS001560View
2D structure for PGDB_C009827
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A015387PGDB_C009827PGDB_AS001560View
2D structure for PGDB_C009811
IC50-=0.5-1uM-—CRBNCRBN-WO2022187423A1PGDB_A016589PGDB_C009811PGDB_AS001560View
2D structure for PGDB_C009828
IC50-=0.5-1uM-—CRBNCRBN-WO2022187423A1PGDB_A017391PGDB_C009828PGDB_AS001560View
2D structure for PGDB_C009799
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A019824PGDB_C009799PGDB_AS001560View
2D structure for PGDB_C009812
IC50-=0.5-1uM-—CRBNCRBN-WO2022187423A1PGDB_A021474PGDB_C009812PGDB_AS001560View
2D structure for PGDB_C009807
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A026965PGDB_C009807PGDB_AS001560View
2D structure for PGDB_C009848
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A029324PGDB_C009848PGDB_AS001560View
2D structure for PGDB_C009801
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A030134PGDB_C009801PGDB_AS001560View
2D structure for PGDB_C009838
IC50-=1-10uM-—CRBNCRBN-WO2022187423A1PGDB_A032086PGDB_C009838PGDB_AS001560View
2D structure for PGDB_C009834
IC50-<=0.5uM-—CRBNCRBN-WO2022187423A1PGDB_A032423PGDB_C009834PGDB_AS001560View
2D structure for PGDB_C009802
IC50-=0.5-1uM-—CRBNCRBN-WO2022187423A1PGDB_A032590PGDB_C009802PGDB_AS001560View
2D structure for PGDB_C009798
IC50->10uM-—CRBNCRBN-WO2022187423A1PGDB_A032719PGDB_C009798PGDB_AS001560View
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