Assay
PGDB_AS001599
System: cell_basedCell line: MDA-MB-436
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.257 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A000425 | PGDB_C030624 | PGDB_AS001599 | View | |
| EC50 | - | = | 0.18 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A002662 | PGDB_C030612 | PGDB_AS001599 | View | |
| EC50 | - | = | 0.312 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A078115 | PGDB_C030609 | PGDB_AS001599 | View | |
| EC50 | - | = | 0.45 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A078372 | PGDB_C030611 | PGDB_AS001599 | View | |
| EC50 | - | = | 1.82 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A079473 | PGDB_C030610 | PGDB_AS001599 | View | |
| EC50 | - | = | 2.47 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A080914 | PGDB_C030622 | PGDB_AS001599 | View |