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Compound
PGDB_C030624
5 activity records1 related patents
2D structure
C[C@H]1CN(c2cc(S(=O)(=O)N(C)C3CC3)cn3c(-c4nnc(C(F)F)s4)nnc23)C[C@H](C)N1C(=O)N(C)CCCCCCCOc1ccc2c(c1)C(=O)N(C1CCC(=O)NC1=O)C2=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.257 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A000425 | PGDB_C030624 | PGDB_AS001599 | View |
| EC50 | - | > | 20 | uM | - | — | PARG | - | U2OS | WO2026062066A1 | PGDB_A001273 | PGDB_C030624 | PGDB_AS002468 | View |
| IC50 | - | = | 0.1 | uM | - | — | PARG | - | - | WO2026062066A1 | PGDB_A006715 | PGDB_C030624 | PGDB_AS002282 | View |
| EC50 | - | = | 0.643 | uM | - | — | PARG | - | NCIH-460 | WO2026062066A1 | PGDB_A078498 | PGDB_C030624 | PGDB_AS002426 | View |
| % Degradation | - | > | 70 | % | - | 0.129 | - | - | MDAMB-436 | WO2026062066A1 | PGDB_A080898 | PGDB_C030624 | PGDB_AS001636 | View |