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Compound
PGDB_C030612
5 activity records1 related patents
2D structure
C[C@H]1CN(c2cc(S(=O)(=O)NC3(C)CC3)cn3c(-c4nnc(C(F)F)s4)ncc23)C[C@H](C)N1C(=O)N1CCC(c2ccc3c(c2)n(C)c(=O)n3C2CCC(=O)NC2=O)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 0.07 | uM | - | — | PARG | - | NCIH-460 | WO2026062066A1 | PGDB_A002392 | PGDB_C030612 | PGDB_AS002426 | View |
| EC50 | - | = | 0.18 | uM | - | — | PARG | - | MDA-MB-436 | WO2026062066A1 | PGDB_A002662 | PGDB_C030612 | PGDB_AS001599 | View |
| IC50 | - | = | 0.093 | uM | - | — | PARG | - | - | WO2026062066A1 | PGDB_A003707 | PGDB_C030612 | PGDB_AS002282 | View |
| % Degradation | - | > | 70 | % | - | 0.129 | - | - | MDAMB-436 | WO2026062066A1 | PGDB_A004045 | PGDB_C030612 | PGDB_AS001636 | View |
| EC50 | - | > | 20 | uM | - | — | PARG | - | U2OS | WO2026062066A1 | PGDB_A005593 | PGDB_C030612 | PGDB_AS002468 | View |