Assay
PGDB_AS001716
System: cell_basedCell line: MDA-MB-231
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 4.7 | nM | - | — | GSPT1 | - | MDA-MB-231 | WO2023001028A1 | PGDB_A039660 | PGDB_C001869 | PGDB_AS001716 | View | |
| IC50 | - | = | 4.7 | nM | - | — | GSPT1 | - | MDA-MB-231 | WO2023001028A1 | PGDB_A053784 | PGDB_C001865 | PGDB_AS001716 | View | |
| IC50 | - | = | 57.2 | nM | - | — | GSPT1 | - | MDA-MB-231 | WO2023001028A1 | PGDB_A055677 | PGDB_C001871 | PGDB_AS001716 | View | |
| IC50 | - | = | 52.4 | nM | - | — | GSPT1 | - | MDA-MB-231 | WO2023001028A1 | PGDB_A056863 | PGDB_C001872 | PGDB_AS001716 | View |