Assay

PGDB_AS001769

System: biochemicalTarget: ALK
Assay context summary

Assay context

129 activity records
Assay familyternary_complex
Systembiochemical
ReadoutFold change
TargetALK
E3CRBN
Activity compounds and values

Activity records

129 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C012278
Emax-=50-120%-2 hALKCRBN-WO2026015344A1PGDB_A008764PGDB_C012278PGDB_AS001769View
2D structure for PGDB_C012389
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A009252PGDB_C012389PGDB_AS001769View
2D structure for PGDB_C012315
Emax-<50%-2 hALKCRBN-WO2026015344A1PGDB_A009634PGDB_C012315PGDB_AS001769View
2D structure for PGDB_C012309
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A010084PGDB_C012309PGDB_AS001769View
2D structure for PGDB_C012336
Emax-<50%-2 hALKCRBN-WO2026015344A1PGDB_A010875PGDB_C012336PGDB_AS001769View
2D structure for PGDB_C012401
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A011921PGDB_C012401PGDB_AS001769View
2D structure for PGDB_C012379
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A012624PGDB_C012379PGDB_AS001769View
2D structure for PGDB_C012363
Emax-<50%-2 hALKCRBN-WO2026015344A1PGDB_A013031PGDB_C012363PGDB_AS001769View
2D structure for PGDB_C012329
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A013050PGDB_C012329PGDB_AS001769View
2D structure for PGDB_C012294
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A013734PGDB_C012294PGDB_AS001769View
2D structure for PGDB_C012305
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A014350PGDB_C012305PGDB_AS001769View
2D structure for PGDB_C012290
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A014459PGDB_C012290PGDB_AS001769View
2D structure for PGDB_C012296
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A014869PGDB_C012296PGDB_AS001769View
2D structure for PGDB_C012277
Emax-=50-120%-2 hALKCRBN-WO2026015344A1PGDB_A014984PGDB_C012277PGDB_AS001769View
2D structure for PGDB_C012461
EC50-=100-1000nM-—ALKCRBN-WO2026015344A1PGDB_A015212PGDB_C012461PGDB_AS001769View
2D structure for PGDB_C012387
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A016320PGDB_C012387PGDB_AS001769View
2D structure for PGDB_C012399
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A016386PGDB_C012399PGDB_AS001769View
2D structure for PGDB_C012473
EC50-=100-1000nM-—ALKCRBN-WO2026015344A1PGDB_A016446PGDB_C012473PGDB_AS001769View
2D structure for PGDB_C012312
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A016510PGDB_C012312PGDB_AS001769View
2D structure for PGDB_C012380
Emax->120%-2 hALKCRBN-WO2026015344A1PGDB_A017919PGDB_C012380PGDB_AS001769View
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