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Compound
PGDB_C012278
4 activity records1 related patents
2D structure
Cc1nc(-c2noc(CN3CCCC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)n2)co1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 50-120 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A008764 | PGDB_C012278 | PGDB_AS001769 | View |
| EC50 | - | = | 100-1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A019576 | PGDB_C012278 | PGDB_AS002152 | View |
| EC50 | - | > | 1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A027451 | PGDB_C012278 | PGDB_AS000738 | View |
| Emax | - | < | 50 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A052502 | PGDB_C012278 | PGDB_AS001094 | View |