Assay
PGDB_AS001781
System: cell_basedCell line: HGC-27
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A009087 | PGDB_C025940 | PGDB_AS001781 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A009611 | PGDB_C025939 | PGDB_AS001781 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A013221 | PGDB_C025948 | PGDB_AS001781 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A016989 | PGDB_C025951 | PGDB_AS001781 | View | |
| IC50 | - | = | 1000-5000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A019883 | PGDB_C016122 | PGDB_AS001781 | View | |
| IC50 | - | = | 100-500 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A024946 | PGDB_C025936 | PGDB_AS001781 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A056799 | PGDB_C025935 | PGDB_AS001781 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A062205 | PGDB_C025950 | PGDB_AS001781 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A064121 | PGDB_C025937 | PGDB_AS001781 | View | |
| IC50 | - | < | 50 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A064775 | PGDB_C025949 | PGDB_AS001781 | View | |
| IC50 | - | = | 500-1000 | nM | - | — | PTK2 | - | HGC-27 | CN116239566A | PGDB_A077346 | PGDB_C025938 | PGDB_AS001781 | View |