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SIMM · NJU
Assay
PGDB_AS001875
System: cell_based
Target: VAV1
Assay context summary
Assay context
190 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
VAV1
E3
Not specified
Technology
luminescence
Detection target
protein_degradation
Activity compounds and values
Activity records
190 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000033
PGDB_C032202
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000104
PGDB_C032078
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000149
PGDB_C032218
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000185
PGDB_C032215
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000243
PGDB_C032115
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000397
PGDB_C032169
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000595
PGDB_C032126
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000606
PGDB_C032164
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000624
PGDB_C032176
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000643
PGDB_C032109
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000685
PGDB_C032213
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000708
PGDB_C032108
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000771
PGDB_C032106
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000798
PGDB_C032124
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000838
PGDB_C032227
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000888
PGDB_C032092
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000891
PGDB_C032211
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A000957
PGDB_C032166
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A001160
PGDB_C032099
PGDB_AS001875
View
DC50
-
<
100
nM
-
—
VAV1
-
-
WO2026119245A1
PGDB_A001193
PGDB_C032237
PGDB_AS001875
View