Assay
PGDB_AS001949
System: cell_basedCell line: A375
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A009173 | PGDB_C011633 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A011980 | PGDB_C011603 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A018805 | PGDB_C011604 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A047681 | PGDB_C011587 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A057134 | PGDB_C011632 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A067277 | PGDB_C011605 | PGDB_AS001949 | View | |
| IC50 | - | > | 1000 | nM | - | — | BRAF | - | A375 | WO2025214350A1 | PGDB_A069532 | PGDB_C011631 | PGDB_AS001949 | View |