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SIMM · NJU
Assay
PGDB_AS002010
System: cell_based
Assay context summary
Assay context
36 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
E3
CRBN
Activity compounds and values
Activity records
36 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
=
288.40315031266056
nM
-
—
-
-
-
EP4683934A1
PGDB_A007451
PGDB_C025571
PGDB_AS002010
View
DC50
-
=
6.309573444801943
nM
-
—
-
-
-
EP4683934A1
PGDB_A014140
PGDB_C025590
PGDB_AS002010
View
DC50
-
=
52.48074602497723
nM
-
—
-
-
-
EP4683934A1
PGDB_A020482
PGDB_C025573
PGDB_AS002010
View
DC50
-
=
12022.644346174131
nM
-
—
-
-
-
EP4683934A1
PGDB_A023418
PGDB_C025581
PGDB_AS002010
View
DC50
-
=
4265.795188015925
nM
-
—
-
-
-
EP4683934A1
PGDB_A024103
PGDB_C025585
PGDB_AS002010
View
DC50
-
=
20.892961308540407
nM
-
—
-
-
-
EP4683934A1
PGDB_A025391
PGDB_C025567
PGDB_AS002010
View
DC50
-
=
107.1519305237607
nM
-
—
-
-
-
EP4683934A1
PGDB_A027185
PGDB_C025566
PGDB_AS002010
View
DC50
-
=
446.6835921509635
nM
-
—
-
-
-
EP4683934A1
PGDB_A028604
PGDB_C025574
PGDB_AS002010
View
DC50
-
=
31.622776601683793
nM
-
—
-
-
-
EP4683934A1
PGDB_A029520
PGDB_C025565
PGDB_AS002010
View
DC50
-
=
21379.620895022323
nM
-
—
-
-
-
EP4683934A1
PGDB_A032216
PGDB_C009602
PGDB_AS002010
View
DC50
-
=
10.232929922807536
nM
-
—
-
-
-
EP4683934A1
PGDB_A034783
PGDB_C025595
PGDB_AS002010
View
DC50
-
=
5754.399373371566
nM
-
—
-
-
-
EP4683934A1
PGDB_A035195
PGDB_C025584
PGDB_AS002010
View
DC50
-
=
14454.39770745928
nM
-
—
-
-
-
EP4683934A1
PGDB_A039324
PGDB_C025583
PGDB_AS002010
View
DC50
-
=
4.3651583224016655
nM
-
—
-
-
-
EP4683934A1
PGDB_A041124
PGDB_C025576
PGDB_AS002010
View
DC50
-
=
3630.78054770101
nM
-
—
-
-
-
EP4683934A1
PGDB_A041673
PGDB_C009602
PGDB_AS002010
View
DC50
-
=
46773.51412871981
nM
-
—
-
-
-
EP4683934A1
PGDB_A041692
PGDB_C025582
PGDB_AS002010
View
DC50
-
=
7.413102413009161
nM
-
—
-
-
-
EP4683934A1
PGDB_A043212
PGDB_C009601
PGDB_AS002010
View
DC50
-
=
3630.78054770101
nM
-
—
-
-
-
EP4683934A1
PGDB_A046948
PGDB_C025572
PGDB_AS002010
View
DC50
-
=
7.943282347242821
nM
-
—
-
-
-
EP4683934A1
PGDB_A047427
PGDB_C025589
PGDB_AS002010
View
DC50
-
=
144.5439770745928
nM
-
—
-
-
-
EP4683934A1
PGDB_A047761
PGDB_C025592
PGDB_AS002010
View