Assay
PGDB_AS002042
System: cell_basedCell line: monocyte-derivedmacrophages
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.108 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A000180 | PGDB_C031217 | PGDB_AS002042 | View | |
| IC50 | - | = | 0.05631 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A002139 | PGDB_C031219 | PGDB_AS002042 | View | |
| IC50 | - | = | 0.008526 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A006364 | PGDB_C031204 | PGDB_AS002042 | View | |
| IC50 | - | = | 0.01261 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A079223 | PGDB_C031225 | PGDB_AS002042 | View | |
| IC50 | - | = | 0.01915 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A079292 | PGDB_C031221 | PGDB_AS002042 | View | |
| IC50 | - | = | 0.2332 | uM | - | — | CASP1 | - | monocyte-derivedmacrophages | WO2026099466A1 | PGDB_A081320 | PGDB_C031230 | PGDB_AS002042 | View |