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SIMM · NJU
Assay
PGDB_AS002057
System: cell_based
Target: IKZF2
Cell line: HEK293
Assay context summary
Assay context
158 activity records
Assay family
% Degradation
System
cell_based
Readout
EC50
Target
IKZF2
E3
Not specified
Cell line
HEK293
Detection target
protein_degradation
Activity compounds and values
Activity records
158 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
0.067
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A009722
PGDB_C005931
PGDB_AS002057
View
EC50
-
=
0.138
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A009898
PGDB_C005996
PGDB_AS002057
View
EC50
-
=
0.042
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A010625
PGDB_C005970
PGDB_AS002057
View
EC50
-
=
0.265
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A010870
PGDB_C005973
PGDB_AS002057
View
EC50
-
=
3.3
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A011058
PGDB_C005905
PGDB_AS002057
View
EC50
-
=
0.171
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A011170
PGDB_C005943
PGDB_AS002057
View
EC50
-
=
0.055
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A011236
PGDB_C005926
PGDB_AS002057
View
EC50
-
=
0.068
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A011881
PGDB_C005982
PGDB_AS002057
View
EC50
-
=
0.525
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A012418
PGDB_C005923
PGDB_AS002057
View
EC50
-
=
1.2
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A013266
PGDB_C005907
PGDB_AS002057
View
EC50
-
=
0.46
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A013390
PGDB_C005920
PGDB_AS002057
View
EC50
-
=
2.8
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A013430
PGDB_C005915
PGDB_AS002057
View
EC50
-
=
0.319
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A013719
PGDB_C005932
PGDB_AS002057
View
EC50
-
=
0.182
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A014418
PGDB_C005914
PGDB_AS002057
View
EC50
-
=
0.003
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A014697
PGDB_C005986
PGDB_AS002057
View
EC50
-
=
1.7
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A014853
PGDB_C005928
PGDB_AS002057
View
EC50
-
=
0.17
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A015096
PGDB_C005993
PGDB_AS002057
View
EC50
-
=
0.588
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A017660
PGDB_C005903
PGDB_AS002057
View
EC50
-
=
0.049
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A018135
PGDB_C005979
PGDB_AS002057
View
EC50
-
=
2
uM
-
—
IKZF2
-
HEK293
AU2022419982A1
PGDB_A018179
PGDB_C005891
PGDB_AS002057
View