Assay context summary

Assay context

77 activity records
Activity compounds and values

Activity records

77 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011631
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A008068PGDB_C011631PGDB_AS002124View
2D structure for PGDB_C028533
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A011023PGDB_C028533PGDB_AS002124View
2D structure for PGDB_C011675
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A011380PGDB_C011675PGDB_AS002124View
2D structure for PGDB_C011623
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A011737PGDB_C011623PGDB_AS002124View
2D structure for PGDB_C028532
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A011807PGDB_C028532PGDB_AS002124View
2D structure for PGDB_C011682
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A013156PGDB_C011682PGDB_AS002124View
2D structure for PGDB_C011614
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A014653PGDB_C011614PGDB_AS002124View
2D structure for PGDB_C011609
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A014680PGDB_C011609PGDB_AS002124View
2D structure for PGDB_C011608
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A014977PGDB_C011608PGDB_AS002124View
2D structure for PGDB_C011596
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A015214PGDB_C011596PGDB_AS002124View
2D structure for PGDB_C011621
IC50->1000nM-KRAS-HPACWO2025214350A1PGDB_A015330PGDB_C011621PGDB_AS002124View
2D structure for PGDB_C011647
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A017387PGDB_C011647PGDB_AS002124View
2D structure for PGDB_C011680
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A017513PGDB_C011680PGDB_AS002124View
2D structure for PGDB_C011646
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A018826PGDB_C011646PGDB_AS002124View
2D structure for PGDB_C011679
IC50-=100-1000nM-KRAS-HPACWO2025214350A1PGDB_A020028PGDB_C011679PGDB_AS002124View
2D structure for PGDB_C011640
IC50-=10-100nM-KRAS-HPACWO2025214350A1PGDB_A020150PGDB_C011640PGDB_AS002124View
2D structure for PGDB_C011619
IC50-=100-1000nM-KRAS-HPACWO2025214350A1PGDB_A022483PGDB_C011619PGDB_AS002124View
2D structure for PGDB_C011685
IC50-=100-1000nM-KRAS-HPACWO2025214350A1PGDB_A022742PGDB_C011685PGDB_AS002124View
2D structure for PGDB_C011645
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A023216PGDB_C011645PGDB_AS002124View
2D structure for PGDB_C011649
IC50-=1-10nM-KRAS-HPACWO2025214350A1PGDB_A024111PGDB_C011649PGDB_AS002124View