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C#Cc1cnc([C@H](C)OC)c(-c2c3c4cc(ccc4n2CC)N2CCC[C@@H](C[C@H](NC(=O)[C@H](C(C)C)N4CC[C@]5(CCN(C(=O)[C@H]6[C@@H](C7CC7)N6C)C5)C4)C(=O)N4N[C@H](C(=O)OCC(C)(C)C3)C3CC4C3)C2)c1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 10-100 | nM | - | — | KRAS | - | AGS | WO2025214350A1 | PGDB_A011693 | PGDB_C011640 | PGDB_AS000218 | View | |
| IC50 | - | = | 10-100 | nM | - | — | KRAS | - | HPAC | WO2025214350A1 | PGDB_A020150 | PGDB_C011640 | PGDB_AS002124 | View | |
| IC50 | - | = | 10-100 | nM | - | — | - | - | AsPC-1 | WO2025214350A1 | PGDB_A055879 | PGDB_C011640 | PGDB_AS001410 | View |