Assay
PGDB_AS002147
System: cell_basedTarget: CCNKCell line: COV362
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 188 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A007569 | PGDB_C006738 | PGDB_AS002147 | View | |
| IC50 | - | = | 10 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A022983 | PGDB_C007161 | PGDB_AS002147 | View | |
| IC50 | - | = | 29 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A034383 | PGDB_C007164 | PGDB_AS002147 | View | |
| IC50 | - | = | 29 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A035214 | PGDB_C007162 | PGDB_AS002147 | View | |
| IC50 | - | = | 28 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A048889 | PGDB_C007160 | PGDB_AS002147 | View | |
| IC50 | - | = | 21 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A052369 | PGDB_C007158 | PGDB_AS002147 | View | |
| IC50 | - | = | 3 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A060286 | PGDB_C007163 | PGDB_AS002147 | View | |
| IC50 | - | > | 1000 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A072257 | PGDB_C007159 | PGDB_AS002147 | View |