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Cn1cc(-n2cnc3c(NCc4nc5cc(Cl)c(Cl)cc5[nH]4)nc(N4CCOCC4)nc32)cn1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 20.28 | nM | - | — | CDK12 | - | MDA-MB-468 | CN121108130A | PGDB_A012172 | PGDB_C007164 | PGDB_AS000556 | View | |
| IC50 | - | = | 7 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A025094 | PGDB_C007164 | PGDB_AS002186 | View | |
| IC50 | - | = | 6 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A031250 | PGDB_C007164 | PGDB_AS002297 | View | |
| IC50 | - | = | 16 | nM | - | — | CCNK | - | SK-OV-3 | CN120329284A | PGDB_A033634 | PGDB_C007164 | PGDB_AS001264 | View | |
| IC50 | - | = | 29 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A034383 | PGDB_C007164 | PGDB_AS002147 | View | |
| IC50 | - | = | 101.28 | nM | - | — | CDK12 | - | - | CN121108130A | PGDB_A062326 | PGDB_C007164 | PGDB_AS002060 | View | |
| IC50 | - | = | 20.75 | nM | - | — | CDK12 | - | MDA-MB-231 | CN121108130A | PGDB_A067450 | PGDB_C007164 | PGDB_AS001069 | View |