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CC[C@H](CO)Nc1nc(NCc2ccc(-c3ccccn3)cc2)c2ncn(C(C)C)c2n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 188 | nM | - | — | CCNK | - | COV362 | CN120329284A | PGDB_A007569 | PGDB_C006738 | PGDB_AS002147 | View | |
| IC50 | - | = | 111 | nM | - | — | CCNK | - | SK-OV-3 | CN120329284A | PGDB_A022503 | PGDB_C006738 | PGDB_AS001264 | View | |
| IC50 | - | = | 53 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A026326 | PGDB_C006738 | PGDB_AS002186 | View | |
| IC50 | - | = | 41 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A048510 | PGDB_C006738 | PGDB_AS002297 | View | |
| IC50 | - | = | 84.5 | nM | - | — | - | - | A673 | JPWO2022263604A5 | PGDB_A064271 | PGDB_C006738 | PGDB_AS002345 | View | |
| IC50 | - | = | 429 | nM | - | — | CCNK | - | HGC-27 | CN117946075A | PGDB_A068407 | PGDB_C006738 | PGDB_AS000524 | View | |
| IC50 | - | = | 302 | nM | - | — | - | - | - | JPWO2022263604A5 | PGDB_A077730 | PGDB_C006738 | PGDB_AS000932 | View |