Assay
PGDB_AS002186
System: cell_basedTarget: CCNKCell line: Jurkat
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 7 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A013073 | PGDB_C007160 | PGDB_AS002186 | View | |
| IC50 | - | = | 11 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A019452 | PGDB_C007162 | PGDB_AS002186 | View | |
| IC50 | - | = | 7 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A025094 | PGDB_C007164 | PGDB_AS002186 | View | |
| IC50 | - | = | 53 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A026326 | PGDB_C006738 | PGDB_AS002186 | View | |
| IC50 | - | = | 1 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A027255 | PGDB_C007163 | PGDB_AS002186 | View | |
| IC50 | - | = | 301 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A032990 | PGDB_C007159 | PGDB_AS002186 | View | |
| IC50 | - | = | 3 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A066860 | PGDB_C007161 | PGDB_AS002186 | View | |
| IC50 | - | = | 2 | nM | - | — | CCNK | - | Jurkat | CN120329284A | PGDB_A074036 | PGDB_C007158 | PGDB_AS002186 | View |