Assay
PGDB_AS002297
System: cell_basedCell line: PA-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A018518 | PGDB_C007161 | PGDB_AS002297 | View | |
| IC50 | - | = | 6 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A031250 | PGDB_C007164 | PGDB_AS002297 | View | |
| IC50 | - | = | 1 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A045415 | PGDB_C007158 | PGDB_AS002297 | View | |
| IC50 | - | = | 148 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A046230 | PGDB_C007159 | PGDB_AS002297 | View | |
| IC50 | - | = | 41 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A048510 | PGDB_C006738 | PGDB_AS002297 | View | |
| IC50 | - | = | 5 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A073064 | PGDB_C007160 | PGDB_AS002297 | View | |
| IC50 | - | = | 4 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A074569 | PGDB_C007162 | PGDB_AS002297 | View | |
| IC50 | - | < | 1 | nM | - | — | CCNK | - | PA-1 | CN120329284A | PGDB_A074627 | PGDB_C007163 | PGDB_AS002297 | View |