Assay context summary

Assay context

31 activity records
Activity compounds and values

Activity records

31 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002563
IC50-=5-10nM---DaudiWO2024032689A1PGDB_A010354PGDB_C002563PGDB_AS002481View
2D structure for PGDB_C002516
IC50-=500-1000nM---DaudiWO2024032689A1PGDB_A011718PGDB_C002516PGDB_AS002481View
2D structure for PGDB_C002557
IC50-=500-1000nM---DaudiWO2024032689A1PGDB_A013924PGDB_C002557PGDB_AS002481View
2D structure for PGDB_C002547
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A023588PGDB_C002547PGDB_AS002481View
2D structure for PGDB_C002534
IC50-=5-10nM---DaudiWO2024032689A1PGDB_A023794PGDB_C002534PGDB_AS002481View
2D structure for PGDB_C002521
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A032863PGDB_C002521PGDB_AS002481View
2D structure for PGDB_C002543
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A036568PGDB_C002543PGDB_AS002481View
2D structure for PGDB_C002533
IC50-=5-10nM---DaudiWO2024032689A1PGDB_A039630PGDB_C002533PGDB_AS002481View
2D structure for PGDB_C002532
IC50-=10-50nM---DaudiWO2024032689A1PGDB_A042964PGDB_C002532PGDB_AS002481View
2D structure for PGDB_C002556
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A043043PGDB_C002556PGDB_AS002481View
2D structure for PGDB_C002565
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A045216PGDB_C002565PGDB_AS002481View
2D structure for PGDB_C002526
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A046117PGDB_C002526PGDB_AS002481View
2D structure for PGDB_C002520
IC50-=500-1000nM---DaudiWO2024032689A1PGDB_A047632PGDB_C002520PGDB_AS002481View
2D structure for PGDB_C002552
IC50-=10-50nM---DaudiWO2024032689A1PGDB_A047652PGDB_C002552PGDB_AS002481View
2D structure for PGDB_C002522
IC50-=500-1000nM---DaudiWO2024032689A1PGDB_A048198PGDB_C002522PGDB_AS002481View
2D structure for PGDB_C002549
IC50-=500-1000nM---DaudiWO2024032689A1PGDB_A051955PGDB_C002549PGDB_AS002481View
2D structure for PGDB_C002498
IC50-=100-500nM---DaudiWO2024032689A1PGDB_A054519PGDB_C002498PGDB_AS002481View
2D structure for PGDB_C002525
IC50-=10-50nM---DaudiWO2024032689A1PGDB_A054952PGDB_C002525PGDB_AS002481View
2D structure for PGDB_C002560
IC50-=50-100nM---DaudiWO2024032689A1PGDB_A056158PGDB_C002560PGDB_AS002481View
2D structure for PGDB_C002564
IC50-=50-100nM---DaudiWO2024032689A1PGDB_A056645PGDB_C002564PGDB_AS002481View