Assay

PGDB_AS001440

System: cell_basedTarget: VAV1
Assay context summary

Assay context

262 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetVAV1
E3Not specified
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

262 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C029684
DC50-=2.3nM-—VAV1--WO2026051943A1PGDB_A000001PGDB_C029684PGDB_AS001440View
2D structure for PGDB_C029462
DC50-=5nM-—VAV1--WO2026051943A1PGDB_A000016PGDB_C029462PGDB_AS001440View
2D structure for PGDB_C029490
DC50-=2.69nM-—VAV1--WO2026051943A1PGDB_A000082PGDB_C029490PGDB_AS001440View
2D structure for PGDB_C029603
DC50-=4.1nM-—VAV1--WO2026051943A1PGDB_A000158PGDB_C029603PGDB_AS001440View
2D structure for PGDB_C029539
DC50-=3.3nM-—VAV1--WO2026051943A1PGDB_A000181PGDB_C029539PGDB_AS001440View
2D structure for PGDB_C029432
DC50-=3.73nM-—VAV1--WO2026051943A1PGDB_A000205PGDB_C029432PGDB_AS001440View
2D structure for PGDB_C029661
DC50-=1.2nM-—VAV1--WO2026051943A1PGDB_A000210PGDB_C029661PGDB_AS001440View
2D structure for PGDB_C029569
DC50-=0.8nM-—VAV1--WO2026051943A1PGDB_A000234PGDB_C029569PGDB_AS001440View
2D structure for PGDB_C029478
DC50-=16.81nM-—VAV1--WO2026051943A1PGDB_A000277PGDB_C029478PGDB_AS001440View
2D structure for PGDB_C029540
DC50-=3.39nM-—VAV1--WO2026051943A1PGDB_A000292PGDB_C029540PGDB_AS001440View
2D structure for PGDB_C029590
DC50-=1.25nM-—VAV1--WO2026051943A1PGDB_A000394PGDB_C029590PGDB_AS001440View
2D structure for PGDB_C029427
DC50-=8.4nM-—VAV1--WO2026051943A1PGDB_A000481PGDB_C029427PGDB_AS001440View
2D structure for PGDB_C029500
DC50-=8.56nM-—VAV1--WO2026051943A1PGDB_A000501PGDB_C029500PGDB_AS001440View
2D structure for PGDB_C029470
DC50-=3.46nM-—VAV1--WO2026051943A1PGDB_A000558PGDB_C029470PGDB_AS001440View
2D structure for PGDB_C029514
DC50-=1.55nM-—VAV1--WO2026051943A1PGDB_A000579PGDB_C029514PGDB_AS001440View
2D structure for PGDB_C029662
DC50-=0.8nM-—VAV1--WO2026051943A1PGDB_A000671PGDB_C029662PGDB_AS001440View
2D structure for PGDB_C029605
DC50-=2.2nM-—VAV1--WO2026051943A1PGDB_A000698PGDB_C029605PGDB_AS001440View
2D structure for PGDB_C029565
DC50-=0.6nM-—VAV1--WO2026051943A1PGDB_A000702PGDB_C029565PGDB_AS001440View
2D structure for PGDB_C029527
DC50-=3.93nM-—VAV1--WO2026051943A1PGDB_A000713PGDB_C029527PGDB_AS001440View
2D structure for PGDB_C029511
DC50-=1.63nM-—VAV1--WO2026051943A1PGDB_A000750PGDB_C029511PGDB_AS001440View
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