Summary
AssigneeGilead Sciences
Filing years2022-2025
Patents4
Compounds517
Activity records2,648
Patent families3
Targets3
Assay familiescellular_function, degradation, viability
Activity metricsDmax, EC50, degradation, fold_change
Overview

Target distribution and active-compound trend

Target distribution

2,648 activity records

3 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

01452892023202420252026
Activity compounds and values

Activity records

2,648 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C005947
Dmax-=67%--IKZF2-HEK293AU2022419982A1PGDB_A007465PGDB_C005947PGDB_AS000473View
2D structure for PGDB_C005897
Dmax-=44%--IKZF1-HEK293AU2022419982A1PGDB_A007700PGDB_C005897PGDB_AS000645View
2D structure for PGDB_C005979
Dmax-=27%--IKZF1-HEK293AU2022419982A1PGDB_A007762PGDB_C005979PGDB_AS000645View
2D structure for PGDB_C005887
Dmax-=95%--IKZF1-HEK293AU2022419982A1PGDB_A007890PGDB_C005887PGDB_AS000645View
2D structure for PGDB_C005956
Dmax-=88%--IKZF1-HEK293AU2022419982A1PGDB_A007912PGDB_C005956PGDB_AS000645View
2D structure for PGDB_C005924
EC50-=0.246uM-IKZF1-HEK293AU2022419982A1PGDB_A007928PGDB_C005924PGDB_AS001788View
2D structure for PGDB_C005976
Dmax-=55%--IKZF1-HEK293AU2022419982A1PGDB_A008074PGDB_C005976PGDB_AS000645View
2D structure for PGDB_C006007
EC50-=0.121uM-IKZF1-HEK293AU2022419982A1PGDB_A008108PGDB_C006007PGDB_AS001788View
2D structure for PGDB_C005952
EC50-=0.07uM-IKZF1-HEK293AU2022419982A1PGDB_A008215PGDB_C005952PGDB_AS001788View
2D structure for PGDB_C005993
Dmax-=85%--IKZF2-HEK293AU2022419982A1PGDB_A008493PGDB_C005993PGDB_AS000473View
2D structure for PGDB_C005965
Dmax-=97%--IKZF2-HEK293AU2022419982A1PGDB_A008546PGDB_C005965PGDB_AS000473View
2D structure for PGDB_C005918
Dmax-=36%--IKZF1-HEK293AU2022419982A1PGDB_A008625PGDB_C005918PGDB_AS000645View
2D structure for PGDB_C005875
EC50-=0.053uM-IKZF1-HEK293AU2022419982A1PGDB_A008818PGDB_C005875PGDB_AS001788View
2D structure for PGDB_C005881
EC50-=0.023uM-IKZF1-HEK293AU2022419982A1PGDB_A008884PGDB_C005881PGDB_AS001788View
2D structure for PGDB_C005934
EC50-=0.07uM-IKZF1-HEK293AU2022419982A1PGDB_A009078PGDB_C005934PGDB_AS001788View
2D structure for PGDB_C006012
EC50-=0.005uM-IKZF1-HEK293AU2022419982A1PGDB_A009136PGDB_C006012PGDB_AS001788View
2D structure for PGDB_C005889
Dmax-=36%--IKZF2-HEK293AU2022419982A1PGDB_A009204PGDB_C005889PGDB_AS000473View
2D structure for PGDB_C005911
EC50-=0.038uM-IKZF1-HEK293AU2022419982A1PGDB_A009210PGDB_C005911PGDB_AS001788View
2D structure for PGDB_C005998
EC50-=0.146uM-IKZF1-HEK293AU2022419982A1PGDB_A009214PGDB_C005998PGDB_AS001788View
2D structure for PGDB_C006006
Dmax-=86%--IKZF2-HEK293AU2022419982A1PGDB_A009513PGDB_C006006PGDB_AS000473View