Summary
AssigneeInnovo Therapeutics
Filing years2023
Patents1
Compounds731
Activity records2,929
Patent families1
Targets2
Assay familiesdegradation
Activity metricsDC50, Ymin
Overview

Target distribution and active-compound trend

Target distribution

3,045 activity records

3 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

03667312025
Activity compounds and values

Activity records

3,045 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C003929
DC50-<25nM-GSPT1-HEK293EP4584259A1PGDB_A007019PGDB_C003929PGDB_AS001862View
2D structure for PGDB_C004143
% Degradation-=0-25%--GSPT1-HEK293EP4584259A1PGDB_A007066PGDB_C004143PGDB_AS001220View
2D structure for PGDB_C004111
DC50-<25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007071PGDB_C004111PGDB_AS001103View
2D structure for PGDB_C003899
% Degradation-=0-25%--GSPT1-HEK293EP4584259A1PGDB_A007094PGDB_C003899PGDB_AS001220View
2D structure for PGDB_C004050
% Degradation-=25-75%--CSNK1A1-HEK293EP4584259A1PGDB_A007116PGDB_C004050PGDB_AS000108View
2D structure for PGDB_C003478
DC50->=25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007139PGDB_C003478PGDB_AS001103View
2D structure for PGDB_C004061
DC50->=25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007178PGDB_C004061PGDB_AS001103View
2D structure for PGDB_C004012
% Degradation-=25-75%--CSNK1A1-HEK293EP4584259A1PGDB_A007181PGDB_C004012PGDB_AS000108View
2D structure for PGDB_C004063
% Degradation-=90-100%-----EP4584259A1PGDB_A007200PGDB_C004063PGDB_AS001586View
2D structure for PGDB_C003698
DC50->=25nM-GSPT1-HEK293EP4584259A1PGDB_A007214PGDB_C003698PGDB_AS001862View
2D structure for PGDB_C003729
% Degradation-=25-75%--CSNK1A1-HEK293EP4584259A1PGDB_A007228PGDB_C003729PGDB_AS000108View
2D structure for PGDB_C003635
DC50->=25nM-GSPT1-HEK293EP4584259A1PGDB_A007229PGDB_C003635PGDB_AS001862View
2D structure for PGDB_C003584
DC50->=25nM-GSPT1-HEK293EP4584259A1PGDB_A007267PGDB_C003584PGDB_AS001862View
2D structure for PGDB_C004057
DC50-<25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007337PGDB_C004057PGDB_AS001103View
2D structure for PGDB_C003625
% Degradation-=0-25%--GSPT1-HEK293EP4584259A1PGDB_A007344PGDB_C003625PGDB_AS001220View
2D structure for PGDB_C003494
DC50->=25nM-GSPT1-HEK293EP4584259A1PGDB_A007361PGDB_C003494PGDB_AS001862View
2D structure for PGDB_C003692
DC50-<25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007389PGDB_C003692PGDB_AS001103View
2D structure for PGDB_C003438
% Degradation-=25-75%--GSPT1-HEK293EP4584259A1PGDB_A007485PGDB_C003438PGDB_AS001220View
2D structure for PGDB_C003564
% Degradation-=0-25%--GSPT1-HEK293EP4584259A1PGDB_A007525PGDB_C003564PGDB_AS001220View
2D structure for PGDB_C003967
DC50-<25nM-CSNK1A1-HEK293EP4584259A1PGDB_A007560PGDB_C003967PGDB_AS001103View