Summary
AssigneeProxygen
Filing years2021-2025
Patents3
Compounds137
Activity records355
Patent families3
Targets1
Assay familiesbinding, degradation, viability
Activity metricsDC50, EC50, LC50
Overview

Target distribution and active-compound trend

Target distribution

444 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

03977202320252026
Activity compounds and values

Activity records

444 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C019114
DC50->10uM-CCNK--AU2021359129A1PGDB_A007396PGDB_C019114PGDB_AS000583View
2D structure for PGDB_C019085
EC50-<=0.25uM---KBM7AU2021359129A1PGDB_A007794PGDB_C019085PGDB_AS000333View
2D structure for PGDB_C019080
LC50-=5.682uM---KBM7AU2021359129A1PGDB_A007968PGDB_C019080PGDB_AS001722View
2D structure for PGDB_C019076
LC50-=1.812uM---KBM7AU2021359129A1PGDB_A008354PGDB_C019076PGDB_AS002507View
2D structure for PGDB_C019083
EC50-=0.5-1uM-CCNK-KBM7AU2021359129A1PGDB_A008519PGDB_C019083PGDB_AS001877View
2D structure for PGDB_C019094
DC50->10uM-CCNK--AU2021359129A1PGDB_A008599PGDB_C019094PGDB_AS000583View
2D structure for PGDB_C019082
DC50-=0.1-0.5uM-CCNK--AU2021359129A1PGDB_A008614PGDB_C019082PGDB_AS000583View
2D structure for PGDB_C019125
DC50-=0.1-0.5uM-CCNK--AU2021359129A1PGDB_A008757PGDB_C019125PGDB_AS000583View
2D structure for PGDB_C019145
DC50-<=0.1uM-CCNK--AU2021359129A1PGDB_A009666PGDB_C019145PGDB_AS000583View
2D structure for PGDB_C019122
EC50->10uM-CCNK-KBM7AU2021359129A1PGDB_A009737PGDB_C019122PGDB_AS001877View
2D structure for PGDB_C019112
EC50-=1-10uM-CCNK--AU2021359129A1PGDB_A010237PGDB_C019112PGDB_AS000733View
2D structure for PGDB_C019118
DC50->10uM-CCNK--AU2021359129A1PGDB_A010272PGDB_C019118PGDB_AS000583View
2D structure for PGDB_C019101
DC50->10uM-CCNK--AU2021359129A1PGDB_A010502PGDB_C019101PGDB_AS000583View
2D structure for PGDB_C019084
DC50->10uM-CCNK--AU2021359129A1PGDB_A010825PGDB_C019084PGDB_AS000583View
2D structure for PGDB_C019134
DC50-=0.1-0.5uM-CCNK--AU2021359129A1PGDB_A011016PGDB_C019134PGDB_AS000583View
2D structure for PGDB_C019139
EC50-=1-10uM-CCNK--AU2021359129A1PGDB_A011506PGDB_C019139PGDB_AS000733View
2D structure for PGDB_C019123
EC50-=0.5-1uM-CCNK--AU2021359129A1PGDB_A011649PGDB_C019123PGDB_AS000733View
2D structure for PGDB_C019143
DC50-<=0.1uM-CCNK--AU2021359129A1PGDB_A012082PGDB_C019143PGDB_AS000583View
2D structure for PGDB_C019127
EC50->10uM-CCNK-KBM7AU2021359129A1PGDB_A012092PGDB_C019127PGDB_AS001877View
2D structure for PGDB_C019136
EC50-=1-10uM-CCNK--AU2021359129A1PGDB_A012463PGDB_C019136PGDB_AS000733View