Summary
AssigneeSuzhou Yasheng Pharmaceutical
Filing years2024
Patents2
Compounds78
Activity records180
Patent families2
Targets1
Assay familiesdegradation, viability
Activity metricsIC50, degradation
Overview

Target distribution and active-compound trend

Target distribution

180 activity records

1 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0255020242025
Activity compounds and values

Activity records

180 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C003233
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A007277PGDB_C003233PGDB_AS002114View
2D structure for PGDB_C003259
% Degradation-=50-80%--GSPT1-KG-1WO2024222918A1PGDB_A007816PGDB_C003259PGDB_AS000482View
2D structure for PGDB_C003232
% Degradation->=80%--GSPT1-KG-1WO2024222918A1PGDB_A008478PGDB_C003232PGDB_AS000482View
2D structure for PGDB_C003263
% Degradation->=80%--GSPT1-KG-1WO2024222918A1PGDB_A011304PGDB_C003263PGDB_AS000482View
2D structure for PGDB_C003239
% Degradation->=80%--GSPT1-KG-1WO2024222918A1PGDB_A011421PGDB_C003239PGDB_AS000482View
2D structure for PGDB_C003222
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A011435PGDB_C003222PGDB_AS002114View
2D structure for PGDB_C003266
IC50-=10-100nM-GSPT1-MOLM-13WO2024222918A1PGDB_A011552PGDB_C003266PGDB_AS000118View
2D structure for PGDB_C003252
% Degradation-=25-50%--GSPT1-KG-1WO2024222918A1PGDB_A011801PGDB_C003252PGDB_AS000482View
2D structure for PGDB_C003237
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A012263PGDB_C003237PGDB_AS002114View
2D structure for PGDB_C003241
% Degradation-=50-80%--GSPT1-KG-1WO2024222918A1PGDB_A012748PGDB_C003241PGDB_AS000482View
2D structure for PGDB_C003249
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A013037PGDB_C003249PGDB_AS002114View
2D structure for PGDB_C003221
IC50-=10-100nM-GSPT1-U937WO2024222918A1PGDB_A014025PGDB_C003221PGDB_AS002362View
2D structure for PGDB_C003228
% Degradation-<25%--GSPT1-KG-1WO2024222918A1PGDB_A015048PGDB_C003228PGDB_AS000482View
2D structure for PGDB_C003236
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A015572PGDB_C003236PGDB_AS002114View
2D structure for PGDB_C003221
IC50-=10-100nM-GSPT1-MOLM-13WO2024222918A1PGDB_A015809PGDB_C003221PGDB_AS000118View
2D structure for PGDB_C000059
IC50-=10-100nM-GSPT1-U937WO2024222918A1PGDB_A016725PGDB_C000059PGDB_AS002362View
2D structure for PGDB_C003262
% Degradation->=80%--GSPT1-KG-1WO2024222918A1PGDB_A018312PGDB_C003262PGDB_AS000482View
2D structure for PGDB_C003238
IC50-=10-100nM-GSPT1-KG-1WO2024222918A1PGDB_A019084PGDB_C003238PGDB_AS002114View
2D structure for PGDB_C003223
IC50-=1-10nM-GSPT1-KG-1WO2024222918A1PGDB_A019248PGDB_C003223PGDB_AS002114View
2D structure for PGDB_C003254
% Degradation->=80%--GSPT1-KG-1WO2024222918A1PGDB_A020984PGDB_C003254PGDB_AS000482View