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Compound
PGDB_C000353
4 activity records1 related patents
2D structure
CC(C)(C)c1ccc(C(=O)NCc2ccc3c(c2)CN(C2CCC(=O)NC2=O)C3=O)cc1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 30-60 | % | 1 uM | - | BRD4 | - | - | CN117683022A | PGDB_A021516 | PGDB_C000353 | PGDB_AS002272 | View |
| IC50 | - | = | 65.9 | nM | - | — | - | - | THP-1 | CN117683022A | PGDB_A035410 | PGDB_C000353 | PGDB_AS000289 | View |
| IC50 | - | = | 54.1 | nM | - | — | - | - | Raji | CN117683022A | PGDB_A061927 | PGDB_C000353 | PGDB_AS000751 | View |
| % Degradation | - | = | 60-80 | % | 1 uM | - | GSPT1 | - | - | CN117683022A | PGDB_A072509 | PGDB_C000353 | PGDB_AS001783 | View |