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Compound
PGDB_C000568
4 activity records2 related patents
2D structure
O=C1CCC(N2Cc3cc(NC(=O)CC4CCN(c5cc(-c6cccc7ccccc67)ccn5)CC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.2 | nM | - | — | - | - | HL-60 | WO2023116835A1 | PGDB_A010145 | PGDB_C000568 | PGDB_AS000718 | View |
| % Degradation | - | = | 77 | % | 10 nM | 24 h | MYC | - | HL-60 | WO2023116835A1 | PGDB_A025079 | PGDB_C000568 | PGDB_AS002563 | View |
| IC50 | - | = | 1.2 | nM | - | — | - | - | HL-60 | CN117982498A | PGDB_A032955 | PGDB_C000568 | PGDB_AS001350 | View |
| % Degradation | - | = | 77 | % | 10 nM | - | - | - | HL-60 | CN117982498A | PGDB_A053717 | PGDB_C000568 | PGDB_AS001270 | View |