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Compound
PGDB_C000589
4 activity records2 related patents
2D structure
O=C1CCC(N2Cc3cc(C(=O)NCC4CCN(c5nccc(-c6ccc7ccccc7c6)n5)CC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 48 | % | 10 nM | - | - | - | HL-60 | CN117982498A | PGDB_A008811 | PGDB_C000589 | PGDB_AS001270 | View |
| IC50 | - | = | 0.9 | nM | - | — | - | - | HL-60 | CN117982498A | PGDB_A065091 | PGDB_C000589 | PGDB_AS001350 | View |
| IC50 | - | = | 0.9 | nM | - | — | - | - | HL-60 | WO2023116835A1 | PGDB_A065328 | PGDB_C000589 | PGDB_AS000718 | View |
| % Degradation | - | = | 48 | % | 10 nM | 24 h | MYC | - | HL-60 | WO2023116835A1 | PGDB_A068840 | PGDB_C000589 | PGDB_AS002563 | View |