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Compound
PGDB_C002015
3 activity records1 related patents
2D structure
O=C1C[C@H](N2Cc3cc(CNCC4CCN(c5ncc(-c6cccc(Cl)c6)cc5C(F)(F)F)CC4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | -5 | % | 10 nM | 24 h | MYC | - | HL-60 | WO2023116835A1 | PGDB_A036904 | PGDB_C002015 | PGDB_AS002563 | View |
| % Degradation | - | = | 35 | % | 10 nM | 24 h | GSPT1 | - | HL-60 | WO2023116835A1 | PGDB_A051109 | PGDB_C002015 | PGDB_AS000871 | View |
| IC50 | - | = | 46.3 | nM | - | — | - | - | HL-60 | WO2023116835A1 | PGDB_A059632 | PGDB_C002015 | PGDB_AS000718 | View |