Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C002258
5 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3cccc(NCc4cccc(C(=O)N[C@H]5CC[C@H](c6nc7cccnc7s6)CC5)c4)c3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 1.48 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A026327 | PGDB_C002258 | PGDB_AS000710 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A035811 | PGDB_C002258 | PGDB_AS001555 | View |
| GI50 | - | = | 1.08 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A044393 | PGDB_C002258 | PGDB_AS002036 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A064573 | PGDB_C002258 | PGDB_AS002200 | View |
| GI50 | - | = | 5.31 | nM | - | — | GSPT1 | - | Raji | WO2023237116A1 | PGDB_A069222 | PGDB_C002258 | PGDB_AS000230 | View |