Assay context summary

Assay context

8 activity records
Activity compounds and values

Activity records

8 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002259
GI50-=5.21nM-GSPT1-NCI-H929WO2023237116A1PGDB_A024168PGDB_C002259PGDB_AS000710View
2D structure for PGDB_C002258
GI50-=1.48nM-GSPT1-NCI-H929WO2023237116A1PGDB_A026327PGDB_C002258PGDB_AS000710View
2D structure for PGDB_C002261
GI50-=7.88nM-GSPT1-NCI-H929WO2023237116A1PGDB_A033868PGDB_C002261PGDB_AS000710View
2D structure for PGDB_C002229
GI50-=1.36nM-GSPT1-NCI-H929WO2023237116A1PGDB_A038872PGDB_C002229PGDB_AS000710View
2D structure for PGDB_C002263
GI50-=0.46nM-GSPT1-NCI-H929WO2023237116A1PGDB_A044045PGDB_C002263PGDB_AS000710View
2D structure for PGDB_C002208
GI50-=6.91nM-GSPT1-NCI-H929WO2023237116A1PGDB_A064180PGDB_C002208PGDB_AS000710View
2D structure for PGDB_C002254
GI50-=0.99nM-GSPT1-NCI-H929WO2023237116A1PGDB_A069795PGDB_C002254PGDB_AS000710View
2D structure for PGDB_C002231
GI50-=2.7nM-GSPT1-NCI-H929WO2023237116A1PGDB_A077528PGDB_C002231PGDB_AS000710View