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Compound
PGDB_C004434
7 activity records1 related patents
2D structure
CC(C)c1ccc(C(=O)C(=O)NCc2scc3c2CN(C2CCC(=O)NC2=O)C3=O)s1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 25-50 | % | 0.1 uM | - | GSPT1 | - | - | US20200369679A1 | PGDB_A025679 | PGDB_C004434 | PGDB_AS001685 | View |
| % Inhibition | - | >= | 80 | % | 1 uM | 3 d | - | - | MOLM-13 | US20200369679A1 | PGDB_A028559 | PGDB_C004434 | PGDB_AS001386 | View |
| % Inhibition | - | >= | 80 | % | 0.1 uM | 1 h | - | - | - | US20200369679A1 | PGDB_A037269 | PGDB_C004434 | PGDB_AS001873 | View |
| % Inhibition | - | >= | 80 | % | 0.1 uM | 24 h | - | - | - | US20200369679A1 | PGDB_A041662 | PGDB_C004434 | PGDB_AS000875 | View |
| % Inhibition | - | >= | 80 | % | 1 uM | 24 h | - | - | - | US20200369679A1 | PGDB_A051274 | PGDB_C004434 | PGDB_AS000693 | View |
| % Inhibition | - | >= | 80 | % | 1 uM | 1 h | - | - | - | US20200369679A1 | PGDB_A066096 | PGDB_C004434 | PGDB_AS000773 | View |
| % Degradation | - | >= | 80 | % | 0.1 uM | - | IKZF1 | - | - | US20200369679A1 | PGDB_A069781 | PGDB_C004434 | PGDB_AS002410 | View |