Assay

PGDB_AS001685

System: cell_basedTarget: GSPT1
Assay context summary

Assay context

6 activity records
Assay family% Degradation
Systemcell_based
Readoutpercent_remaining
TargetGSPT1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

6 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C004431
% Degradation-=50-80%0.1 uM-GSPT1--US20200369679A1PGDB_A013044PGDB_C004431PGDB_AS001685View
2D structure for PGDB_C004434
% Degradation-=25-50%0.1 uM-GSPT1--US20200369679A1PGDB_A025679PGDB_C004434PGDB_AS001685View
2D structure for PGDB_C004435
% Degradation->=80%0.1 uM-GSPT1--US20200369679A1PGDB_A026459PGDB_C004435PGDB_AS001685View
2D structure for PGDB_C004432
% Degradation->=80%0.1 uM-GSPT1--US20200369679A1PGDB_A049600PGDB_C004432PGDB_AS001685View
2D structure for PGDB_C004436
% Degradation-=50-80%0.1 uM-GSPT1--US20200369679A1PGDB_A058893PGDB_C004436PGDB_AS001685View
2D structure for PGDB_C004433
% Degradation-=50-80%0.1 uM-GSPT1--US20200369679A1PGDB_A064889PGDB_C004433PGDB_AS001685View
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