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Compound
PGDB_C004436
4 activity records1 related patents
2D structure
Cc1ccc(NC(=O)NCc2cc3c(s2)C(=O)N(C2CCC(=O)NC2=O)C3)cc1N(C)CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 25-50 | % | 1 uM | 1 h | - | - | - | US20200369679A1 | PGDB_A009129 | PGDB_C004436 | PGDB_AS000773 | View |
| % Inhibition | - | >= | 80 | % | 1 uM | 3 d | - | - | MOLM-13 | US20200369679A1 | PGDB_A039814 | PGDB_C004436 | PGDB_AS001386 | View |
| % Degradation | - | = | 50-80 | % | 0.1 uM | - | GSPT1 | - | - | US20200369679A1 | PGDB_A058893 | PGDB_C004436 | PGDB_AS001685 | View |
| % Inhibition | - | = | 25-50 | % | 1 uM | 24 h | - | - | - | US20200369679A1 | PGDB_A076336 | PGDB_C004436 | PGDB_AS000693 | View |