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Compound
PGDB_C005363
3 activity records1 related patents
2D structure
Cc1ncc(NC(=O)OCc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3)cc1C#CC1CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Degradation | - | = | 3.41 | % | Concentration context: 100 nM | 6 h | GSPT1 | - | NCI-H1155 | WO2024125437A1 | PGDB_A008992 | PGDB_C005363 | PGDB_AS001010 | View |
| % Degradation | - | = | 30.46 | % | Concentration context: 10 nM | 6 h | GSPT1 | - | NCI-H1155 | WO2024125437A1 | PGDB_A011864 | PGDB_C005363 | PGDB_AS000061 | View |
| IC50 | - | = | 4.2 | nM | - | — | - | - | NCI-H1155 | WO2024125437A1 | PGDB_A073753 | PGDB_C005363 | PGDB_AS001656 | View |