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Compound
PGDB_C005730
2 activity records1 related patents
2D structure
CCN(CC)S(=O)(=O)c1cc(F)c(Oc2ccc3ncn([C@H]4COC5(CCN(C(=O)CN6CCC(c7ccc(NC8CCC(=O)NC8=O)cc7F)CC6)CC5)C4)c(=O)c3c2Cl)c(C#N)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 31.78 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A014744 | PGDB_C005730 | PGDB_AS001091 | View |
| Emax | - | = | 9.51 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A053233 | PGDB_C005730 | PGDB_AS000014 | View |