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Compound
PGDB_C005763
2 activity records1 related patents
2D structure
CO[C@H]1CCN(S(=O)(=O)Nc2ccc(F)c(Oc3ccc4ncn(-c5cnc(N6CCN(C(=O)CN7CCC(c8ccc(N[C@H]9CCC(=O)NC9=O)cc8F)CC7)CC6)nc5)c(=O)c4c3)c2C#N)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 10.27 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A017638 | PGDB_C005763 | PGDB_AS001074 | View |
| DC50 | - | = | 18.62 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A023197 | PGDB_C005763 | PGDB_AS001629 | View |