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Compound
PGDB_C005771
2 activity records1 related patents
2D structure
CN(CC(F)F)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn(-c4cnc(N5CCN(C(=O)CN6CCC(c7ccc(N[C@@H]8CCC(=O)NC8=O)cc7F)CC6)CC5)nc4)c(=O)c3c2)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 12.8 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A018113 | PGDB_C005771 | PGDB_AS001074 | View |
| DC50 | - | = | 46.91 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A050684 | PGDB_C005771 | PGDB_AS001629 | View |