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Compound
PGDB_C005848
2 activity records1 related patents
2D structure
CN(C1CC1)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn([C@@H]4CC5(CCN(C(=O)CC6(O)CCN(c7cc8c(cc7F)c(N7CCC(=O)NC7=O)nn8C)CC6)CC5)O4)c(=O)c3c2)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 27.76 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A014825 | PGDB_C005848 | PGDB_AS000362 | View |
| DC50 | - | = | 25.7 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A054485 | PGDB_C005848 | PGDB_AS001308 | View |