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Compound
PGDB_C005854
2 activity records1 related patents
2D structure
CCN(C)S(=O)(=O)Nc1ccc(F)c(Oc2ccc3ncn([C@H]4COC5(CCN(C(=O)CN6CC[C@H](c7cc8c(cc7F)c(N7CCC(=O)NC7=O)nn8C)C(F)(F)C6)CC5)C4)c(=O)c3c2)c1C#NCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | = | 11.27 | % | 10 uM | 24 h | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A011288 | PGDB_C005854 | PGDB_AS000362 | View |
| DC50 | - | = | 37.53 | nM | - | — | BRAF | - | A375.10 | AU2022290851A1 | PGDB_A052738 | PGDB_C005854 | PGDB_AS001308 | View |