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CCn1cnc2c(NCc3nc4cc(Cl)c(Cl)cc4[nH]3)nc(N3CCN(C(=O)c4cccnc4)CC3)nc21| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 14.12 | nM | - | — | CDK12 | - | MDA-MB-231 | CN120590389A | PGDB_A018166 | PGDB_C007245 | PGDB_AS000401 | View | |
| IC50 | - | = | 2.411 | nM | - | — | CDK12 | - | MDA-MB-468 | CN120590389A | PGDB_A063793 | PGDB_C007245 | PGDB_AS000658 | View |