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CCCCOc1nc(NCc2nc3cc(Cl)c(Cl)cc3[nH]2)c2ncn(CC)c2n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 122.9 | nM | - | — | CDK12 | - | MDA-MB-468 | CN120590389A | PGDB_A045340 | PGDB_C007273 | PGDB_AS000658 | View | |
| IC50 | - | = | 199 | nM | - | — | CDK12 | - | MDA-MB-231 | CN120590389A | PGDB_A061528 | PGDB_C007273 | PGDB_AS000401 | View |