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CC(=O)N1CCN(c2nc(NCc3nc4cc(Cl)c(Cl)cc4[nH]3)c3ncn(C)c3n2)CC1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 153.3 | nM | - | — | CDK12 | - | MDA-MB-231 | CN120590389A | PGDB_A047938 | PGDB_C007285 | PGDB_AS000401 | View | |
| IC50 | - | = | 82.05 | nM | - | — | CDK12 | - | MDA-MB-468 | CN120590389A | PGDB_A058673 | PGDB_C007285 | PGDB_AS000658 | View |