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Cn1cc(-n2cnc3c(NCc4nc5cc(Cl)c(Cl)cc5[nH]4)nc(N4CCNCC4)nc32)cn1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 15.68 | nM | - | — | CDK12 | - | MDA-MB-468 | CN120590389A | PGDB_A044847 | PGDB_C007286 | PGDB_AS000658 | View | |
| IC50 | - | = | 63.8 | nM | - | — | CDK12 | - | MDA-MB-231 | CN120590389A | PGDB_A062083 | PGDB_C007286 | PGDB_AS000401 | View |